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Mankhwala "stugeron" malangizo Buku.

Mankhwala "stugeron": The mawonekedwe kumasulidwa, kapangidwe ndi wazolongedza

Mapiritsi woyera, mosabisa, kuzungulira, ndi mbali imodzi, ndi pafupifupi palibe fungo kumbali imodzi - mawu akuti "STUGERON", mamiligalamu twente-faifi wa pophika yogwira - cinnarizine, matuza pa magome twente-faifi ndi makumi asanu. The zikuchokera zikuphatikizapo, kuwonjezera cinnarizine, ndi zambiri adjuvants: colloidal silika, wowuma mbatata, magnesium stearate, talc, povidone, wowuma chimanga, lactose monohydrate.

Zotsatira pharmacological wa mankhwala "stugeron" malangizo Buku limafotokoza njira zotsatirazi.

Amachepetsa otaya ayoni kashiamu m'zipinda, kamvekedwe ka ulusi yosalala minofu m'makoma arterioles, timapitiriza zotsatira ulesi ziwiya mpweya woipa ndi zambiri. Chifukwa mankhwala "stugeron" zotsatira mwachindunji minofu mtima yosalala, ndi anachepetsa kubvomereza kwawo kwa michere (Epinephrine, angiotensin, dopamine, vasopressin). Iwo ali zotsatira vasodilating (makamaka okhudza ziwiya oziziritsa), koma alibe chikoka kwambiri pa mtengo magazi. Akusonyeza antihistaminic ntchito amakhudza dongosolo vestibular, kucheperachepera excitability ake, ndi chifundo mantha dongosolo, kutsitsa kamvekedwe ake. Kumachititsanso kuwonjezeka mu elasticity erythrocyte Kakhungu ndi luso lawo deform, kuchepetsa magazi kukhuthala. Komanso, minofu ya thupi kumawonjezera kukaniza kuti hypoxia.

The pharmacokinetics wa mankhwala "stugeron" malangizo ntchito anafotokoza choncho.

Resorption mankhwala akupezeka matumbo ndi m'mimba. Ndende pazipita mu madzi pambuyo utsogoleli wa mankhwala mkati Zimapezeka ndi chimodzi - maola atatu. plasma mapuloteni kumumanga ndi nainte imodzi cinnarizine. Metoboliziruet kukonzekera (by glyukuronirovaniya) kwathunthu mu chiwindi. theka moyo wake nthawi ndi maola anayi. Metabolites tsinnarizina linanena bungwe ndi gawo limodzi mwa impso, ndi kulandilidwa ndi mphambu ziwili za intestine ndi.

Mlingo wa Buku mankhwala "stugeron" malangizo amapereka zotsatirazi.

Landira ayenera, pambuyo chakudya. Pamene oziziritsa magazi matenda - twente-faifi - mamiligalamu makumi asanu (imodzi - mapiritsi awiri) katatu patsiku. Pamene zotumphukira magazi matenda - makumi asanu - mamiligalamu makumi asanu (awiri - mapiritsi atatu) katatu patsiku. Ndipo mu nkhani ya matenda vestibular - chifukwa mamiligalamu twente-faifi (piritsi limodzi) katatu patsiku. Pamene "njira" ya matenda (kinetoses) - mlingo akuluakulu - chifukwa mamiligalamu twente-faifi, theka la ola pamaso ulendo (ngati n'koyenera, ayenera kutenga maola monga mmene zisanu), "stugeron" ana Zikatero, kupereka pa theka mlingo akuluakulu. Mu nkhani ya hypersensitivity mmodzi wa zigawo zikuluzikulu za mankhwala "stugeron" malangizo Buku akulimbikitsidwa kuyamba mankhwala ndi theka la mlingo, pang'onopang'ono kuwonjezeka izo. The njira ya mankhwala zambiri kumatenga kwa milungu ingapo. The pazipita kololeka tsiku mlingo "stugeron" malangizo Buku amapereka mamiligalamu mazana asanu kapena miyala naini.

Pankhaniyi cha mankhwala osokoneza bongo - kuwawa m'mimba kusamba madzi abwino, kupereka adamulowetsa makala.

Ndipo ngati mankhwala Kwalamulidwa "stugeron" ana?

Ndemanga pa maukonde ikukhudzana makamaka udindo wake ndi perinatal encephalopathy akuwuka kwa hypoxia yoopsa, komanso ndi perinatal CNS chotupa ndi matenda a neuro-reflex excitability. Linanena ena zotsatira zabwino. Zotchulidwa dokotala nadzam'ninkha anayi la piritsi kawiri pa tsiku mukatha kudya, grinded mu supuni ndi osakaniza kudyetsa kapena kumapeto kwa kudya. Kumapeto - kupereka zotsalira chakumwa Kusakaniza kapena madzi.

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