Mapangidwe, Sayansi
Pamene kutumikiridwa tetracycline. malangizo
Tetracycline kuchitira pharmacological gulu la zinthu la dzina chomwecho. Mu maonekedwe ake angwiro ndi crystalline ufa wa chikasu, odorless, kulawa zowawa. Iwo akusonyeza mphamvu otsika kupasuka osati madzi komanso mowa. Sitichedwa kuvunda mu zidulo amphamvu ndi alkalis. Hygroscopic. Ngati yaitali kukhudzana ndi kuwala amamuchititsa mdima.
The kanthu pharmacological wa tetracycline akhoza zimachitika sipekitiramu wothandizila akuluakulu antibacterial, izo akusonyeza chuma bacteriostatic. Tetracycline amachititsa chisokonezo mapangidwe kuipidwa pakati pa ribosome ndi mayendedwe a RNA, izo zimabweretsa chisokonezo mu ndondomeko ya kaphatikizidwe mapuloteni. Iye akugwira ntchito ndi yaikulu mndandanda wa galamu mabakiteriya, tizilombo galamu HIV, mogwira amalimbana ndi chiwerengero cha tizilombo tina.
Koma palinso mndandanda wa tizilombo kuti ndi kugonjetsedwa ndi mankhwala. Amafuna kuchipatala pamaso kumwa mankhwala okhala ndi tetracycline. Guide amapereka zambiri yekha ndipo si chiongoko kudzimvera mankhwala.
Mbali ya nkhaniyi okha, 75-77% kuchuluka mlingo wa suction, amene nawonso amakhudza kudya chakudya ndi kapangidwe kake. Mankhwala anatengedwa pamaso chakudya, makamaka ngati chakudya pali mkaka, imatsala woipa kuposa chopanda kanthu m'mimba. Zotsatira achire kumachitika pamene thupi mu ndende zina, monga ulamuliro, zimenezi zimafuna masiku 2-3 ya ingestion zonse.
Tetracycline akusonyeza kwambiri malowedwe luso mu zimakhala zosiyana ndi ziwalo, madzi a m'thupi. Iwo akhoza kudziunjikira mu mafupa, ndulu, chiwindi, zotupa, mano. Wakutheker kugonjetsa nsengwa ndi kulowa mkaka mayi. thunthu ndi nthawi yaitali mu thupi la munthu. Pa tsiku loyamba maola 12 a impso anali mwayeretsa chamoyo wa tetracycline chifukwa 10-20% ya mlingo. Gawo la mlingo mu kuchuluka kwa 5-10% ya okwana ndi ya ndulu mu intestine, koma pano mwina tsankho suction, ndi thunthu tikalowa m'thupi kumbuyo.
Tetracycline ali zikuonetsa ntchito matenda opatsirana. Ndi chibayo ndi matenda thirakiti kupuma , iye anasankhidwa kuti mkati. Mankhwala odzola okhala ndi tetracycline, malangizo ntchito kulengeza ntchito mankhwala ndi ziphuphu zakumaso vulgaris ndi matenda bakiteriya khungu. A wapadera diso mafuta ( "Akos Tetracycline") zochokera mankhwala ntchito pa matenda oyamba ndi bakiteriya ocular. Muli ya tetracycline m'maso.
mankhwala ambiri dzina lawo, mwachitsanzo, "amafunika tetracycline-Lect." Uzani zambiri, kuchuluka uli tetracycline, malangizo aliyense mankhwala enieni.
Sitiyenera kuiwala zigawo "contraindications" ndi "mavuto." Musati kumwa tetracycline malangizo pa wachiwiri ndi wachitatu trimester mimba, pa mkaka wa m'mawere, ndi ana kwa zaka 8. Chenjezo kusamala ngati hypersensitivity ntchito mafuta ndi madontho. Nthawi zina pa phwando tetratsiklinsoderzhaschih mankhwala angakhalepo zochita zoipa.
Izi akhoza kusonyeza kuti utachepa kudya, pakutchulidwa kuchita nseru, kusanza, kutsekula m'mimba, glossitis, gastritis, esophagitis, chapamimba predyazvennogo boma 12 mmatumbo chilonda; maonekedwe a hypertrophy a chinenero papillae, chifuwa ndi zochita immunopathological ndi mavuto ena osafunika. Mulimonsemo, kuwonongeka kwa boma ambiri thanzi chifukwa cha ntchito mankhwala aliwonse ayenera kuonana ndi dokotala. Makamaka m'pofunika kupewa kudzikonda mankhwala, ngakhale kukhalapo ngakhale chiongoko bwino ndi zambiri mu mawonekedwe a malangizo.
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